Previous edition: 2008.
Section 1 – General Aspects of Medicinal Chemistry
Section 2 – Lead Compound Discovery Strategies
Section 3 – Primary Exploration of Structure-Activity Relationships
Section 4 – Substituents and Functions: Qualitative and Quantitative Aspects of Structure-Activity Relationships
Section 5 – Spatial Organization, Receptor Mapping and Molecular Modeling
Section 6 – Chemical Modifications Influencing the Pharmacokinetic Properties
Section 7 – Pharmaceutical and Chemical Means to Solubility and Formulation Problems
The practice of medicinal chemistry. ISBN 9780124172135. Published by Academic Press in 2015. Publication and catalogue information, links to buy online and reader comments.